Date of Award

2026

Document Type

Open Access Master's Thesis

Degree Name

Master of Science in Chemistry (MS)

Administrative Home Department

Department of Chemistry

Advisor 1

Tarun Dam

Committee Member 1

Smitha Rao-Hatti

Committee Member 2

Lynn R. Mazzoleni

Abstract

Glycosides, a group of clinically important plant-derived natural products, can kill a wide variety of cells (including pathogens and cancer cells) by disrupting cell membranes. Structurally, a glycoside contains a hydrophobic core, which is covalently linked to one or more sugar (monosaccharide) molecules. Glycosides are generally hemolytic, meaning they lyse (disintegrate) red blood cells (RBCs). Therefore, hemolysis assays using rabbit or human RBC are performed to identify glycosides and to measure their activity. Despite their clinical importance, most plant glycosides are difficult to purify. This thesis describes the isolation and purification of a new glycoside from a monocot plant by using an activity-guided fractionation workflow. The glycoside in crude mixture was extracted from the plant tissues with methanol. The methanol extract was separated by solvent partitioning by using organic solvents and water. The water layer was dried and was subjected to chromatographic separation techniques including P100 size exclusion chromatography (SEC), thin layer chromatography (TLC), silica-gel chromatography and HPLC. After separation, structural analysis was done by MALDI-MS and ESI-MS. The separated glycoside has a mass (m/z) of 1737 Da. ESI spectra and acid hydrolysis data indicate that the glycoside is composed of a core aglycone and several structural sugars. Ligand binding property and thermal stability of the glycoside were also determined and its hemolytic effects on red blood cells were documented by scanning electron microscopy (SEM). The important discovery of a new glycoside, as described in this thesis, sets the stage for future studies for assessing the antimicrobial and anticancer properties of this new bioactive compound.

Available for download on Wednesday, June 09, 2027

Included in

Chemistry Commons

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