Title

Psilocin analogs II. Synthesis of 3‐[2‐(dialkylamino)ethyl]‐, 3‐[2‐(N‐methyl‐N‐alkylamino)ethyl]‐, and 3‐[2‐(cycloalkylamino)ethyl]indol‐4‐ols

Document Type

Article

Publication Date

1-1-1981

Abstract

Structural alteration of the Nb‐substituents of psilocin (3‐[2‐dimethylamino)ethyl]indol‐4‐ol) (12a) has led to a number of compounds containing known pharmacophoric groups. Further, it is hoped that the subtle changes in the nature of these substituents may lead to a clearer understanding of the structure‐activity relationships of the 4‐hydroxytryptamine hallucinogens. Copyright © 1981 Journal of Heterocyclic Chemistry

Publication Title

Journal of Heterocyclic Chemistry

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